Not Tribulus terrestris, but Tribulus alatus (over 600mg in T-Anabol)
Tribulus alatus is a plant that grows in the Sahara and Middle East. It is a relative of Tribulus terrestris, well known in the sports world in the form of supplements which manufacturers claim raise testosterone levels. Recent studies have put paid to these claims, but according to Egyptian researchers, T. alatus is a different kettle of fish.
The Egyptians did tests on male rats. The animals were given extracts of Tribulus alatus through a tube into the stomach every day for a period of forty days. Afterwards the researchers measured the amount of free testosterone in the rats’ blood.
Tribulas Alatus:
Investigative Urology Tribulus Alatus Extracts and Testosterone Level
International Braz J Urol Vol. 33 (4): 554-559, July - August, 2007
Free Serum Testosterone Level in Male Rats Treated with
Tribulus Alatus Extracts
Walid H. El-Tantawy, Abeer Temraz, Omayma D. El-Gindi
Drug Bioavailability Center, National Organization For Drug Control and Research, Cairo, Egypt,
Pharmacognosy Department, Faculty of Pharmacy for Girls, Al-Azhar University, Cairo, Egypt
ABSTRACT
Objective: The present study was undertaken to investigate the effect of Tribulus alatus extracts on free serum testosterone
in male rats.
Materials and Methods: Free serum testosterone level was measured in male rats treated with alcoholic extracts of the
aerial part without fruits, fruits of Tribulus alatus and their fractions.
Results: All tested extracts showed significant increase in the level of free serum testosterone when compared to that of
corresponding control, p < 0.05. Statistical comparison of all groups revealed that the maximum level was found in groups
treated with chloroformic and ethanolic fractions of fruits extract.
Conclusion: Tribulus alatus extract appears to possess aphrodisiac activity due to its androgen increasing property.
Key words: Tribulus; testosterone; aphrodisiacs; rats
Int Braz J Urol. 2007; 33: 554-9
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What is Equipoise?
It is a favorite veterinary steroid of many athletes. Its effects are strongly anabolic, and only moderately androgenic. By itself, Boldagen will provide a steady and consistent gain in mass and strength. However, best results are achieved when Equipoise is used in conjunction with other steroids.
Equipoise is a favorite veterinary steroid of many athletes. Its effects are strongly anabolic, and only moderately androgenic. By itself, Boldagen will provide a steady and consistent gain in mass and strength. However, best results are achieved when Boldagen is used in conjunction with other steroids.For mass, Boldagen stacks exceptionally well with Methanoplex, Oxyplex or an injectable testosterone like Sustaplex 325or Testaplex C. Equipoise is also highly effective for contest preparation since it aromatizes very poorly. Muscle hardness and density can be greatly improved when Equipoise is combined with Enanthate or Winstrol.
What is Glucophage?
Glucophage is an oral antidiabetic medication used to treat type 2 (non-insulin-dependent) diabetes. Diabetes develops when the body proves unable to burn sugar and the unused sugar builds up in the bloodstream. Glucophage lowers the amount of sugar in your blood by decreasing sugar production and absorption and helping your body respond better to its own insulin, which promotes the burning of sugar. It does not, however, increase the body"s production of insulin.
Glucophage was made to be used to control adult onset diabetes. This drug is will increase the body"s ability to transport glucose into the muscle cells much better by increasing insulin sensitivity. This substance will also inhibit the body"s formation of sugar by the liver whereby lowering insulin secretion in the body. This substance is very similar to phenformin that is also an oral hypoglycemic except that phenformin is considered the harsher of the two compounds. Phenformin is considered to be from 5 - 10 times stronger than Glucophage at what it does for the body on a mg. per mg. comparison. Glucophage has signifigantly less side effects than phenformin has as well. The chance for an overdose causing hypoglycemia with the use of Glucophage is dose related whereas you almost have to take a lethal dose. It is common knowledge that Glucophage will increase insulin sensitivity as well. As far as bodybuilders are concerned, this product is used as an oral form of insulin. It will cause greater glycogen supercompensation during carb-ups as well as lowering blood glucose for those that are using the BodyOpus or Atkins diet to induce ketosis more easily. Common side effects of Glucophage are a metallic taste in the mouth, nausea, and vomiting. This will become on the next big drugs used by professional bodybuilders in the coming years for its ability as a repartitioning agent and blood glucose disposal agent.
Whats Andriol?
Andriol is one of the few new steroids developed during the last few years. Unlike most anabolic steroids which were found on the market during the 1950"s and 1960"s (and which in part, have disappeared) Andriol has only been available since the early 1980"s. This fact probably explains why Andriol holds a special place among the steroids. Andriol is a revolutionary steroid because, besides methyltestosterone, it is the only effective oral testosterone compound. Testosterone itself, if taken orally, is ineffective since it is reabsorbed through the portal vein and immediately deactivated by the liver. How it worksThe substance testosterone undecanoate contained in Andriol, however, is reabsorbed from the intestine through the lymphatic system, thus bypassing the liver and becoming effective. The liver function is not affected by this. Testosterone undecanoate is a fatty acid ester of the natural androgen, testosterone, and in the body is for the most part transformed into dihydrotestosterone, a metabolite of testosterone. For this reason Andriol aromatizes only minimally, meaning that only a very small part of the substance can be converted into estrogen, since the dihydrotestosterone does not aromatize. The users of Andriol therefore do not experience feminization symptoms such as gynecomastia or increased body fat.This makes it a welcome alternative for athletes who have problems with the common injectable testosterone compounds. Due to this, Andriol is also suitable for pre competition workouts. An additional advantage of Andriol is non-aromatizing quality consists of the fact that the body"s own hormone production is only affected after a long-term administration of very high dosages. Andriol has only a low inhibitive effect on the hypothalamus so that the release of LHRH (luteinizing hormone releasing hormone) is rarely influenced. This is very important since-as we know-LHRH stimulates the hypophysis to release gonadotropine which causes the Ledig"s cells in the testes to produce testosterone. Consequently, Andriol should be the perfect steroid; however, this is not the case.Side effectsThe disadvantage of Andriol is that it becomes effective if taken in high doses. Even if a dose of 200 mg of Andriol/day is taken, the testosterone level in the blood is still too low for a bodybuilder to gain strength and muscle growth. The need for such a high daily dosage can be explained by its extremely short half-life time since the substance testosterone undecanoate is excreted very quickly by the body through the urine. The capsules, therefore, are effective for only a few hours so that 6-7 capsules, that is 240-280 mg (minimum), must be taken daily to achieve good results comparable to those of injectable compounds. This, however, puts the athlete in a dosage range which begins to influence the hormone production and the compound now more readily converts into estrogen. Such a dose can also manifest itself in a higher retention of sodium and water. This is one factor which competing athletes must consider. DosagesAnother disadvantage is Andriol"s high price. For those athletes who would like to try Andriol 8 capsules ( 320 mg daily) should be taken. The capsules should be taken three times daily (approximately every 8 hours) after meals so that the substance can be properly reabsorbed. However, even this high dosage does not guarantee satisfactory results. Those of you who believe that you need even higher doses should then consider that it might be more sensible to switch to the injectable testosterone. Andriol is often combined with Anavar since Anavar also does not suppress the production of testosterone and, in addition, does not aromatize. The Andriol/Anavar stack gives athletes who do not yet have much experience with steroids a fairly large strength increase and also often substantial muscle growth. For athletes over forty this combination is also of interest. Those working out for competitions and wanting to avoid injections on a regular basis can substitute Testosterone propionate with Andriol. Women and AndriolSince Andriol is quickly eliminated by the body it should also be considered for use before competitions requiring doping tests. Women should avoid Andriol since the androgenic component common with testosterone is also strongly developed in this compound. Andriol intake can occasionally lead to high blood pressure, retention of fluids, acne, sexual over stimulation, and, in women, the well known virilization symptoms.The greatest advantage of Andriol lies in its good compatibility. It can, for example, be used with Deca Durabolin in long-term therapy and, in this combination and for health-conscientious athletes, it is an alternative to the famous Dianabol (D-bol)/Deca Durabolin stack. Theoretically, Andriol should build up muscle and mass, in combination with noticeable water retention, in a fast and reliable way, similar to the tested injectable Testosterone Sustanon and Testoviron Depot. Unfortunately, this is not the case. Some athletes who work out for a competition store too much water due to their use of the injectable testosterone, resulting in smooth muscles. However, if they still do not want to give up Testo, they should at least not have the estrogen-linked complications caused by taking up to 240 mg Andriol/day and be able to reduce the water retention. In this phase, the estrogen level must be kept as low as possible, otherwise the best diet will be useless. The intake of Andriol makes sense in this case and usually brings acceptable results. Otherwise, Andriol is a drug better used by hobby-bodybuilders.
Sleep Well
A good 7-8 hours of uninterrupted sleep is a must for our body to reboot itself and feel energetic next day. Lack of sleep affects our hormone levels and slows down metabolism often resulting in weight gain. Studies have shown that deep, uninterrupted sleep helps cell growth and cell repair, which can increase the metabolism and help in burning calories.
Whats HGH ?
The use of exogenous sources of Growth Hormone has been popular in the United States for almost 8 years now. Originally, athletes used biologically active forms that were the actual extract of the pituitary glands of cadavers. While production was under way on the synthetic, recombinant DNA versions of this drug, it was discovered that the biologically active form was associated with the formation of a rare brain virus called Creutzveldt Jacob Disease. This was a fatal virus that afflicted a very small number of GH users, none of whom were athletes. In light of this discovery, the FDA removed all of these natural GH versions from the market in the United States. Luckily, the synthetic recombinant versions were approved by the FDA a short time afterwards. These versions were developed after years of experiments with amino acid chains. The first of these versions was patented and produced by Genentech Labs with the brand name Protropin. A short time later, another form of synthetic Growth Hormone gained FDA approval. It was produced by Eli Lilly Labs and brand named Humatrope. This product was allowed to be patented because it was shown to be unique in that it contained a slightly different amino acid chain than the Protropin. The difference was that Humatrope had 191 amino acid chains in sequence and Protropin had 192. For some very complicated reasons, the 191 amino acid configuration has been shown to be more effective. It had been speculated that these synthetic versions of GH would greatly improve the cost effectiveness of using GH, yet that has not been the case.�It has been used extensively by athletes who are attempting to alter their body composition. Growth Hormone itself, is an endogenous hormone produced by the pituitary gland. It exists at especially high levels during the teen years when it promotes growth of almost all tissues. It also contributes to the deposition of protein and promotes the breakdown of fat for use as energy. As the body reaches full maturation, the endogenous levels of GH are substantially diminished. After this, GH is still present in the body but at a substantially lower level where it continues to aid in protein synthesis, RNA and DNA reactions and the conversion of body fat to energy. By introducing an exogenous source of this hormone, athletes are hoping to promote these effects, causing the body to deposit more muscle tissue while atthe same time reducing body fat stores. On paper, GH should work exceptionally well; however, it does not seem to be delivering up to its potential. Most athletes who have experimented with this product end up being disappointed. There is some evidence that exogenous sources of GH are being destroyed by antibodies which appear after the introduction of the synthetic compound. Although the 191 amino acid sequence versions have been shown to produce less of an antibody reaction, they are still not yielding consistent results. I have speculated as to whether the introduction of exogenous GH would yield an appreciable degree of efficacy simply due to the fact that the body does not have sufficient receptor affinity to GH in the post-teen years. A number of athletes claim that GH is not that effective on its own, but in a stack with steroids it can do remarkable things. Perhaps there is some type of actual synergism created by the concomitant use of these two agents. Empirical data suggests that the efficacy of GH is dose related and that the majority of users may not have been taking enough Although Growth Hormone is banned by athletic committees, there is no method for the detection of it which allows drug tested competitors to use this product freely without any ramifications. Adverse reactions to GH use are rare but technically could involve a cromegaly (elongation of the feet, forehead and hands). Other possible side effects involve overgrowth of the elbows or jaw, thickening of the skin and a type of diabetes. Effective dosages seem to be in the area of 4 IU/day. Cycle length is usually determined by how long the athlete can afford it. Some take the product for 6 week cycles, others use it year round
Whats Insulin ?
Insulin is a powerful hormone in the human body, responsible for regulating glucose levels in the blood. This is a function that your life constantly depends on. Before going any further I must stress that insulin use by those who do not medically require it can be a very risky endeavor. It is important not only to research and understand the risks involved, but to really give some thought to just how important a little extra boost is to you. Misusing insulin can have tragic results. Immediate death, coma or the possible development of insulin dependent diabetes in a previously healthy athlete are all possible, be extremely careful.
In the human body insulin is secreted by the pancreas. The release of this hormone is most closely tied to glucose, although a number of other factors including pancreatic & gastrointestinal hormones, amino acids, fatty acids and ketone bodies are also involved. Its role in the body is to control the uptake, utilization and storage of amino acids, carbohydrates and fatty acids by various cells of your body. The activity of insulin is both anabolic and anti-catabolic, the hormone stimulating the use and retention cellular nutrients while inhibiting their breakdown. Skeletal muscle cells are among the many targets of this hormone’s action, and the reason pharmaceutical insulin has made its way into the realm of athletics. But this is a little tricky because insulin can also promote nutrient storage in fat cells, obviously an unwanted result. Athletes have found however, that a strict regimen of intense weight training and a diet without excess caloric intake can result in insulin showing a much higher affinity for protein and carbohydrate storage in muscle cells. This could produce rapid and noticeable growth, the muscles beginning to look fuller (and sometimes more defined) almost immediately after starting insulin therapy.